Abstract |
|
Authors | Giulio Auciello, Annalise Di Marco, Odalys Gonzalez Paz, Savina Malancona, Steven Harper, Maria Beconi, Ilaria Rossetti, Alina Ciammaichella, Paola Fezzardi, Andrea Vecchi, Elena Bracacel, Daniel Cicero, Edith Monteagudo, Daniel Elbaum |
Journal | Journal of medicinal chemistry
(J Med Chem)
Vol. 63
Issue 24
Pg. 15785-15801
(12 24 2020)
ISSN: 1520-4804 [Electronic] United States |
PMID | 33320012
(Publication Type: Journal Article)
|
Chemical References |
- Prodrugs
- Pantothenic Acid
- phosphopantothenic acid
- Coenzyme A
|
Topics |
- Animals
- Blood-Brain Barrier
(drug effects, metabolism)
- Brain
(metabolism)
- Coenzyme A
(metabolism)
- Cyclization
- Disease Models, Animal
- Half-Life
- Hepatocytes
(cytology, metabolism)
- Humans
- Lipid Droplets
(chemistry, metabolism)
- Mice
- Mice, Inbred C57BL
- Mice, Knockout
- Pantothenate Kinase-Associated Neurodegeneration
(drug therapy, pathology)
- Pantothenic Acid
(analogs & derivatives, chemistry, metabolism, therapeutic use)
- Prodrugs
(chemistry, metabolism, therapeutic use)
- Structure-Activity Relationship
|