Abstract |
|
Authors | Ahmed Morsy, Paul C Trippier |
Journal | ACS chemical biology
(ACS Chem Biol)
Vol. 15
Issue 3
Pg. 646-650
(03 20 2020)
ISSN: 1554-8937 [Electronic] United States |
PMID | 32125151
(Publication Type: Journal Article, Research Support, N.I.H., Extramural)
|
Chemical References |
- Androgen Antagonists
- Antineoplastic Agents
- Benzamides
- Enzyme Inhibitors
- Nitriles
- Pyrazoles
- Thiohydantoins
- apalutamide
- darolutamide
- Phenylthiohydantoin
- enzalutamide
- Aldo-Keto Reductase Family 1 Member C3
- Prostate-Specific Antigen
|
Topics |
- Aldo-Keto Reductase Family 1 Member C3
(genetics, metabolism)
- Androgen Antagonists
(metabolism)
- Antineoplastic Agents
(metabolism)
- Benzamides
- Cell Line, Tumor
- Cell Proliferation
(drug effects)
- Drug Discovery
- Drug Resistance, Neoplasm
(drug effects)
- Drug Therapy, Combination
- Enzyme Inhibitors
(metabolism)
- Gene Expression Regulation
(drug effects)
- Humans
- Male
- Nitriles
- Orchiectomy
- Phenylthiohydantoin
(analogs & derivatives, metabolism)
- Prostate-Specific Antigen
(metabolism)
- Prostatic Neoplasms, Castration-Resistant
(drug therapy)
- Pyrazoles
(metabolism)
- Substrate Specificity
- Thiohydantoins
(metabolism)
|