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N- (4- chloro- 3- methoxyphenyl)- 2- picolinamide
a positive allosteric modulator of mGlu4 receptor
Also Known As:
ML128 compound; N-(4-chloro-3-(11C)methoxyphenyl)-2-picolinamide; VU0361737
Networked:
1
relevant articles (
0
outcomes,
0
trials/studies)
Bio-Agent Context: Research Results
Organic Chemicals: 133
Amines: 4871
Aniline Compounds: 46
N-(4-chloro-3-methoxyphenyl)-2-picolinamide: 1
Heterocyclic Compounds: 198
1-Ring Heterocyclic Compounds
Pyridines: 88
Picolinic Acids: 1
N-(4-chloro-3-methoxyphenyl)-2-picolinamide: 1
Heterocyclic Acids
Picolinic Acids: 1
N-(4-chloro-3-methoxyphenyl)-2-picolinamide: 1
Experts
1.
Greda, A
: 1 article (09/2015)
2.
Grygier, B
: 1 article (09/2015)
3.
Jantas, D
: 1 article (09/2015)
4.
Lason, W
: 1 article (09/2015)
5.
Leskiewicz, M
: 1 article (09/2015)
6.
Pilc, A
: 1 article (09/2015)
Related Diseases
1.
Neuroblastoma
09/01/2015 - "
Thus, the comparison of the neuroprotective potency of the mGluR II agonist LY354740, mGluR III agonist ACPT-I, mGluR4 PAM VU0361737, mGluR8 PAM AZ12216052 and allosteric mGluR7 agonist AMN082 against staurosporine (St-) and doxorubicin (Dox)-induced cell death has been performed in undifferentiated (UN-) and retinoic acid differentiated (RA-) human neuroblastoma SH-SY5Y cells.
"
Related Drugs and Biologics
1.
Staurosporine
2.
Tretinoin (Retinoic Acid)
3.
Doxorubicin (Adriamycin)
4.
AZ 12216052
5.
N,N'-dibenzhydrylethane-1,2-diamine dihydrochloride
6.
metabotropic glutamate receptor 8
7.
metabotropic glutamate receptor 4
8.
1-aminocyclopentane-1,3,4-tricarboxylic acid
9.
eglumetad
10.
metabotropic glutamate receptor 7