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PLX7904
a RAF inhibitor; structure in first source
Also Known As:
5-(2-cyclopropylpyrimidin-5-yl)-3-(3-((ethyl(methyl)sulfamoyl)amino)-2,6-difluorobenzoyl)-1H-pyrrolo(2,3-b)pyridine
Networked:
1
relevant articles (
0
outcomes,
0
trials/studies)
Bio-Agent Context: Research Results
Heterocyclic Compounds: 198
Fused-Ring Heterocyclic Compounds
2-Ring Heterocyclic Compounds
PLX7904: 1
Organic Chemicals: 133
Amides: 2428
Sulfonamides: 2809
PLX7904: 1
Sulfur Compounds: 278
Sulfones: 534
Sulfonamides: 2809
PLX7904: 1
Experts
1.
Aplin, Andrew E
: 1 article (05/2014)
2.
Basile, Kevin J
: 1 article (05/2014)
3.
Hartsough, Edward J
: 1 article (05/2014)
4.
Le, Kaitlyn
: 1 article (05/2014)
Related Diseases
1.
Melanoma (Melanoma, Malignant)
05/01/2014 - "
Next-generation RAF inhibitors, such as PLX7904 (PB04), effectively inhibit RAF signaling in BRAF(V600E) melanoma cells without paradoxical effects in wild-type cells.
"